EMT Inhibitor-2, targeting both CYP3A4 testosteron and CYP2C9, exhibits inhibitory effects with IC50 values of 49.72 and 5.54 µM, respectively. Furthermore, it effectively impedes the epithelial-mesenchymal transition (EMT) process, induced by immunocyte-released agents like IL-1beta and TGF-beta.
Molekulargewicht:
470.47
CAS Nummer:
[2232228-60-1]
Formel:
C24H26N2O8
Target-Kategorie:
Cytochromes P450|||Others
T11187
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