FGTI-2734, CAS [[1247018-19-4]]

Artikelnummer: TGM-T11282
Artikelname: FGTI-2734, CAS [[1247018-19-4]]
Artikelnummer: TGM-T11282
Hersteller Artikelnummer: T11282
Alternativnummer: TGM-T11282-1MLX10MM(INDMSO), TGM-T11282-1MG, TGM-T11282-5MG, TGM-T11282-10MG, TGM-T11282-25MG, TGM-T11282-50MG, TGM-T11282-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
FGTI-2734 is a dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT-1) inhibitor, exhibiting IC50 values of 250 nM and 520 nM for FT and GGT-1, respectively. It effectively prevents the membrane localization of KRAS, addressing the issue of KRAS resistance and inhibiting the growth of mutant KRAS patient-derived pancreatic tumors.
Molekulargewicht: 510.63
Reinheit: 99.36%
CAS Nummer: [1247018-19-4]
Formel: C26H31FN6O2S
Target-Kategorie: Ras|||Transferase|||Kras
T11282