Samidorphan hydrochloride is an orally active opioid system modulator that has a high affinity for binding with µ-opioid, kappa-opioid, and delta-opioid receptors. Samidorphan hydrochloride acts as an antagonist at µ-opioid receptors and acts as a partial agonist at k-opioid and delta-opioid receptors. Samidorphan hydrochloride primarily acts as an opioid receptor antagonist in vivo. Samidorphan can improve the behavior of depressed animals[1].
Molecular Weight:
406.90
CAS Number:
[2328045-02-7]
Formula:
C21H27ClN2O4
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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