Androgen receptor antagonist 12, CAS [[6605-17-0]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-169349
Supplier Catalog Number:
HY-169349
Alternative Catalog Number:
MCE-HY-169349-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Androgen receptor antagonist 12 (Compound EF2) is an orally active Androgen receptor (AR) antagonist (IC50: 0.30 µM). Androgen receptor antagonist 12 inhibits transcriptional activity of variant AR mutants and and the proliferation of AR-positive PCa cell lines. Androgen receptor antagonist 12 blocks AR nuclear translocation. Androgen receptor antagonist 12 inhibits tumor growth in a C4-2B xenograft mouse model. Androgen receptor antagonist 12 can be used for prostate cancer (PCa) research[1].
Molecular Weight:
283.21
CAS Number:
[6605-17-0]
Formula:
C12H8F3N3O2
Target:
Androgen Receptor
Application Notes:
Reference compound
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