Androgen receptor antagonist 12, CAS [[6605-17-0]] Preis auf Anfrage

Catalog Number: MCE-HY-169349
Article Name: Androgen receptor antagonist 12, CAS [[6605-17-0]] Preis auf Anfrage
Biozol Catalog Number: MCE-HY-169349
Supplier Catalog Number: HY-169349
Alternative Catalog Number: MCE-HY-169349-1UNIT
Manufacturer: MedchemExpress
Category: Biochemikalien
Androgen receptor antagonist 12 (Compound EF2) is an orally active Androgen receptor (AR) antagonist (IC50: 0.30 µM). Androgen receptor antagonist 12 inhibits transcriptional activity of variant AR mutants and and the proliferation of AR-positive PCa cell lines. Androgen receptor antagonist 12 blocks AR nuclear translocation. Androgen receptor antagonist 12 inhibits tumor growth in a C4-2B xenograft mouse model. Androgen receptor antagonist 12 can be used for prostate cancer (PCa) research[1].
Molecular Weight: 283.21
CAS Number: [6605-17-0]
Formula: C12H8F3N3O2
Target: Androgen Receptor
Application Notes: Reference compound