Arg-IN-1 is a selective Arginine (Arg)-targeting covalent inhibitor with IC50s of 9.7 nM and 30.4 nM for FGFR2 and FGFR3,respectively. Arg-IN-1 has the potential to avoid FGFR1/4-targeted toxicity as well as conquer acquired on-target resistance, potential for FGFR-targeting cancer therapy[1].
Molecular Weight:
738.80
Formula:
C36H42N12O6
Target:
FGFR
Application Notes:
MCE Product type: Reference compound
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