GR-4991W93 is an orally active partial agonist against 5HT1B/1D receptor, with pIC50 values of 6.95 and 7.80 against 5HT1B and 5HT1D, respectively. GR-4991W93 demonstrates potent inhibition of electrically evoked plasma extravasation in the guinea pig. GR-4991W93 can be used for migraine research[1].
Molecular Weight:
313.39
CAS Number:
[171549-56-7]
Formula:
C18H23N3O2
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound
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