EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 µM) against human EP1, EP2, and EP3 receptors.
Molecular Weight:
458.43
Purity:
99.53%
CAS Number:
[2287259-07-6]
Formula:
C23H21F3N4O3
Target:
Prostaglandin Receptor
T11211
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