Bazedoxifene (TSE-424) is an oral, BBB-penetrant nonsteroidal selective estrogen receptor modulator (SERM), with IC50s of 23 nM and 99 nM for ERalpha and ERbeta, respectively. Bazedoxifene also acts as an inhibitor of IL-6/GP130 protein-protein interactions and can be used for the research of pancreatic cancer.
Molekulargewicht:
470.6
Reinheit:
>98.50%
CAS Nummer:
[198481-32-2]
Formel:
C30H34N2O3
Target-Kategorie:
Estrogen Receptor
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