Clobenpropit dihydrobromide, CAS [[145231-35-2]]

Artikelnummer: AMO-M28480
Artikelname: Clobenpropit dihydrobromide, CAS [[145231-35-2]]
Artikelnummer: AMO-M28480
Hersteller Artikelnummer: M28480
Alternativnummer: AMO-M28480-5MG,AMO-M28480-10MG,AMO-M28480-25MG,AMO-M28480-50MG
Hersteller: Abmole Bioscience
Kategorie: Biochemikalien
Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors (Ki 7.4 nM) and alpha2A/alpha2C adrenoceptors (Ki 17.4/7.8 nM). Clobenpropit dihydrobromide increases apoptosis.
Molekulargewicht: 470.65
Reinheit: 99.0%
CAS Nummer: [145231-35-2]
Formel: C14H19Br2ClN4S
Target-Kategorie: Histamine Receptor