Samuraciclib, CAS [[1805833-75-3]]

Artikelnummer: AMO-M28894
Artikelname: Samuraciclib, CAS [[1805833-75-3]]
Artikelnummer: AMO-M28894
Hersteller Artikelnummer: M28894
Alternativnummer: AMO-M28894-5MG,AMO-M28894-10MG
Hersteller: Abmole Bioscience
Kategorie: Biochemikalien
Alternative Synonym: CT7001, ICEC0942
Samuraciclib (CT7001) is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 µM. Samuraciclib has anti-tumor effects.
Molekulargewicht: 394.51
Reinheit: 98.0%
CAS Nummer: [1805833-75-3]
Formel: C22H30N6O
Target-Kategorie: CDK