GSK215, CAS [[2743427-26-9]]

Artikelnummer: AMO-M29789
Artikelname: GSK215, CAS [[2743427-26-9]]
Artikelnummer: AMO-M29789
Hersteller Artikelnummer: M29789
Alternativnummer: AMO-M29789-5MG,AMO-M29789-10MG,AMO-M29789-25MG,AMO-M29789-50MG
Hersteller: Abmole Bioscience
Kategorie: Biochemikalien
GSK215 is a potent and selective PROTAC focal adhesion kinase (FAK) degrader with a pDC50 of 8.4. GSK215 is designed by a binder for the VHL E3 ligase and the FAK inhibitor VS-4718. GSK215 induces rapid and prolonged FAK degradation, giving a long-lasting effect on FAK levels and a marked pharmacokinetic/pharmacodynamics (PK/PD) disconnect.
Molekulargewicht: 985.13
Reinheit: 99.0%
CAS Nummer: [2743427-26-9]
Formel: C50H59F3N10O6S
Target-Kategorie: FAK