Deucravacitinib (BMS-986165), CAS [[1609392-27-9]]
Artikelnummer:
AMO-M4138
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| Artikelname: | Deucravacitinib (BMS-986165), CAS [[1609392-27-9]] |
| Artikelnummer: | AMO-M4138 |
| Hersteller Artikelnummer: | M4138 |
| Alternativnummer: | AMO-M4138-1MG,AMO-M4138-5MG,AMO-M4138-10MG,AMO-M4138-25MG |
| Hersteller: | Abmole Bioscience |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | BMS986165 |
| Deucravacitinib (BMS-986165) is a first-in-class, selective, orally bioavailable inhibitor of TYK2 transitions.Deucravacitinib selectively binds the TYK2 pseudokinase (JH2) structural domain with an IC50 of 1.0 nM and a Ki value of 0.02 nM. Deucravacitinib (BMS-986165) blocks receptor-mediated Tyk2 activation by stably regulating the JH2 structural domain. deucravacitinib also inhibits the IL-12/23 and type I IFN pathways. deucravacitinib may be used in psoriasis research. |
| Molekulargewicht: | 425.46 |
| Reinheit: | 99.17% |
| CAS Nummer: | [1609392-27-9] |
| Formel: | C20H19D3N8O3 |
| Target-Kategorie: | JAK |
