Deucravacitinib (BMS-986165), CAS [[1609392-27-9]]

Artikelnummer: AMO-M4138
Artikelname: Deucravacitinib (BMS-986165), CAS [[1609392-27-9]]
Artikelnummer: AMO-M4138
Hersteller Artikelnummer: M4138
Alternativnummer: AMO-M4138-1MG,AMO-M4138-5MG,AMO-M4138-10MG,AMO-M4138-25MG
Hersteller: Abmole Bioscience
Kategorie: Biochemikalien
Alternative Synonym: BMS986165
Deucravacitinib (BMS-986165) is a first-in-class, selective, orally bioavailable inhibitor of TYK2 transitions.Deucravacitinib selectively binds the TYK2 pseudokinase (JH2) structural domain with an IC50 of 1.0 nM and a Ki value of 0.02 nM. Deucravacitinib (BMS-986165) blocks receptor-mediated Tyk2 activation by stably regulating the JH2 structural domain. deucravacitinib also inhibits the IL-12/23 and type I IFN pathways. deucravacitinib may be used in psoriasis research.
Molekulargewicht: 425.46
Reinheit: 99.17%
CAS Nummer: [1609392-27-9]
Formel: C20H19D3N8O3
Target-Kategorie: JAK