Alvimopan dihydrate, CAS [[170098-38-1]]
Artikelnummer:
AMO-M5403
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| Artikelname: | Alvimopan dihydrate, CAS [[170098-38-1]] |
| Artikelnummer: | AMO-M5403 |
| Hersteller Artikelnummer: | M5403 |
| Alternativnummer: | AMO-M5403-5MG,AMO-M5403-10MG,AMO-M5403-50MG |
| Hersteller: | Abmole Bioscience |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | LY 246736 dihydrate, ADL 8-2698 dihydrate |
| Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible µ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for µ-opioid receptor (Ki=0.47 nM) over kappa- and delta-opioid receptors (Kis=100, 12 nM, respectively). |
| Molekulargewicht: | 460.56 |
| Reinheit: | >98.5% |
| CAS Nummer: | [170098-38-1] |
| Formel: | C25H36N2O6 |
| Target-Kategorie: | Opioid Receptor |
