BMS-986365 (CC-94676) is a selective heterobifunctional ligand-directed degrader (LDD) with a dual mechanism-of-action and best-in-class potential, targeting the androgen receptor (AR). In animal models of advanced prostate cancer, BMS-986365 demonstrates on-target activity, degrading AR, suppressing AR signaling, and inhibiting tumor growth.
Molekulargewicht:
818.91
Reinheit:
>99.0%
CAS Nummer:
[2446928-30-7]
Formel:
C41H45F3N8O5S
Target-Kategorie:
Androgen Receptor
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