IDH2-C100, IHD2 Inhibitor, CAS [[1446506-78-0]], Unconjugated

Artikelnummer: BSS-BS-60190C
Artikelname: IDH2-C100, IHD2 Inhibitor, CAS [[1446506-78-0]], Unconjugated
Artikelnummer: BSS-BS-60190C
Hersteller Artikelnummer: bs-60190C
Alternativnummer: BSS-BS-60190C-10,BSS-BS-60190C-2
Hersteller: Bioss
Kategorie: Biochemikalien
Konjugation: Unconjugated
IDH2-C100 is a potent and selective inhibitor of IDH2 R140Q and R172K mutant first reported in patent WO 2013102431. It can inhibit the enzymatic activity of IDH2 R140Q and R172K in vitro with an IC50 < 0.1 µM. It has IC50 < 0.1 µM in U87MG pLVX-IDH2 R140Q-neo cell based assay. It is an analog of clinical IDH2 inhibitor AG-221 by Thomson Reuters Integrity analysis.
Puffer: Powder
CAS Nummer: [1446506-78-0]