CFTR Inhibitor II(GlyH101), CAS [[328541-79-3]], Unconjugated
Artikelnummer:
BSS-BS-6419C
Hersteller Artikelnummer:
bs-6419C
Alternativnummer:
BSS-BS-6419C-10,BSS-BS-6419C-2
Hersteller:
Bioss
Kategorie:
Biochemikalien
Konjugation:
Unconjugated
CFTR Inhibitor II is a CFTR inhibitor (cystic fibrosis transmembrane conductance regulator). CFTR Inhibitor II is a glycine hydrazide that has been shown to block CFTR channels. CFTR Inhibitor II blocked I(Cl.PKA) in a concentration- and voltage-dependent fashion (IC(50) at +100 mV=0.3 1.5 µM and at -100 mV=5.1 1.3 µM). CFTR Inhibitor II blocks the open pore of cardiac CFTR channels at an electrical distance of 0.15 0.03 from the external membrane surface.
Puffer:
Powder
CAS Nummer:
[328541-79-3]
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