PLX51107, CAS [[1627929-55-8]]

Artikelnummer: BYT-ORB1296097
Artikelname: PLX51107, CAS [[1627929-55-8]]
Artikelnummer: BYT-ORB1296097
Hersteller Artikelnummer: orb1296097
Alternativnummer: BYT-ORB1296097-1, BYT-ORB1296097-1, BYT-ORB1296097-10, BYT-ORB1296097-100, BYT-ORB1296097-2, BYT-ORB1296097-25, BYT-ORB1296097-5, BYT-ORB1296097-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: BET, inhibit, PLX 51107, PLX51107, PLX-51107, Inhibitor, EpigeneticReaderDomain, Epigenetic Reader Domain
PLX51107 is a potent, selective BET bromodomain inhibitor with low nanomolar affinity for BRD2, BRD3, BRD4, and BRDT. This small molecule is a valuable research tool for investigating BET protein function in oncology, immunology, and inflammation, supporting both in vitro biochemical assays and in vivo preclinical studies.
Molekulargewicht: 438.48
Reinheit: 99.75% (May vary between batches)
CAS Nummer: [1627929-55-8]
Formel: C26H22N4O3
Target-Kategorie: Epigenetic Reader Domain
Anwendungsbeschreibung: Solubility: DMSO:70 mg/mL (159.64 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.56 mM)