Derazantinib, CAS [[1234356-69-4]]
Artikelnummer:
BYT-ORB1296116
Produktübersicht
Artikelname:
Derazantinib, CAS [[1234356-69-4]]
Artikelnummer:
BYT-ORB1296116
Hersteller Artikelnummer:
orb1296116
Alternativnummer:
BYT-ORB1296116-1, BYT-ORB1296116-1, BYT-ORB1296116-10, BYT-ORB1296116-100, BYT-ORB1296116-200, BYT-ORB1296116-25, BYT-ORB1296116-5, BYT-ORB1296116-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
ARQ 087, ARQ087, ARQ-087, Derazantinib, inhibit, Inhibitor, Fibroblast growth factor receptor, FGFR, FGFR1, FGFR2, FGFR3
Produktbeschreibung
Derazantinib (ARQ-087) is an orally bioavailable, ATP-competitive inhibitor targeting fibroblast growth factor receptors (FGFRs) with low nanomolar potency. It is used in research to investigate FGFR-driven pathologies, demonstrating activity in both in vitro assays and in vivo tumor models.
Produkteigenschaften
Molekulargewicht:
468.57
Reinheit:
99.95% (May vary between batches)
CAS Nummer:
[1234356-69-4]
Formel:
C29H29FN4O
Target-Kategorie:
FGFR
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (7.04 mM),DMSO:98 mg/mL (209.15 mM)