NI-57, CAS [[1883548-89-7]]

Artikelnummer: BYT-ORB1296217
Artikelname: NI-57, CAS [[1883548-89-7]]
Artikelnummer: BYT-ORB1296217
Hersteller Artikelnummer: orb1296217
Alternativnummer: BYT-ORB1296217-1, BYT-ORB1296217-10, BYT-ORB1296217-2, BYT-ORB1296217-25, BYT-ORB1296217-5, BYT-ORB1296217-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: BRPF1, BRPF2, BRPF3, inhibit, Inhibitor, NI 57, NI57, NI-57, EpigeneticReaderDomain, Epigenetic Reader Domain
NI-57 is a potent small molecule inhibitor targeting the BRPF family of proteins, exhibiting IC50 values of 3.1 nM for BRPF1, 46 nM for BRPF2/BRD1, and 140 nM for BRPF3. This compound is a valuable chemical probe for epigenetic research, enabling the investigation of BRPF function in chromatin regulation and gene expression in both cellular and biochemical assays.
Molekulargewicht: 383.42
Reinheit: >99.99% (May vary between batches)
CAS Nummer: [1883548-89-7]
Formel: C19H17N3O4S
Target-Kategorie: Epigenetic Reader Domain
Anwendungsbeschreibung: Solubility: DMSO:80 mg/mL (208.65 mM),10% DMSO+90% Corn Oil:3.3 mg/mL (8.61 mM)