MI-503, CAS [[1857417-13-0]]

Artikelnummer: BYT-ORB1296227
Artikelname: MI-503, CAS [[1857417-13-0]]
Artikelnummer: BYT-ORB1296227
Hersteller Artikelnummer: orb1296227
Alternativnummer: BYT-ORB1296227-1, BYT-ORB1296227-1, BYT-ORB1296227-10, BYT-ORB1296227-100, BYT-ORB1296227-25, BYT-ORB1296227-5, BYT-ORB1296227-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: MI 503, MI503, MI-503, Inhibitor, inhibit, Epigenetic Reader Domain, EpigeneticReaderDomain, Menin-MLL, Histone Methyltransferase, HistoneMethyltransferase
MI-503 is a potent and selective Menin-MLL interaction inhibitor exhibiting an IC50 of 14.7 nM. It demonstrates significant anti-proliferative activity in human MLL-rearranged leukemia cell lines with GI values ranging from 250 to 570 nM, supporting its use in both in vitro and in vivo cancer research.
Molekulargewicht: 564.63
Reinheit: 99.99% (May vary between batches)
CAS Nummer: [1857417-13-0]
Formel: C28H27F3N8S
Target-Kategorie: Epigenetic Reader Domain,Histone Methyltransferase
Anwendungsbeschreibung: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.54 mM),DMSO:45 mg/mL (79.7 mM),H2O:Insoluble