Fadraciclib, CAS [[1070790-89-4]]

Artikelnummer: BYT-ORB1296241
Artikelname: Fadraciclib, CAS [[1070790-89-4]]
Artikelnummer: BYT-ORB1296241
Hersteller Artikelnummer: orb1296241
Alternativnummer: BYT-ORB1296241-1, BYT-ORB1296241-1, BYT-ORB1296241-10, BYT-ORB1296241-100, BYT-ORB1296241-2, BYT-ORB1296241-25, BYT-ORB1296241-5, BYT-ORB1296241-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: CDK9, CDK, CDK2, Cyclin dependent kinase, CYC 065, CYC065, CYC-065, inhibit, Fadraciclib, Inhibitor
Fadraciclib (CYC065) is a potent, orally bioavailable inhibitor targeting CDK2 and CDK9 kinases with IC50 values of 5 nM and 26 nM, respectively. It is used in cancer research to study transcriptional regulation and apoptosis, demonstrating activity in both in vitro cell-based assays and in vivo tumor models.
Molekulargewicht: 397.52
Reinheit: 99.75% (May vary between batches)
CAS Nummer: [1070790-89-4]
Formel: C21H31N7O
Target-Kategorie: CDK
Anwendungsbeschreibung: Solubility: DMSO:100 mg/mL (251.56 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (10.06 mM)