TGFbetaRI-IN-3, CAS [[2763602-67-9]]
Artikelnummer:
BYT-ORB1298043
Produktübersicht
Artikelname:
TGFbetaRI-IN-3, CAS [[2763602-67-9]]
Artikelnummer:
BYT-ORB1298043
Hersteller Artikelnummer:
orb1298043
Alternativnummer:
BYT-ORB1298043-1, BYT-ORB1298043-1, BYT-ORB1298043-10, BYT-ORB1298043-100, BYT-ORB1298043-25, BYT-ORB1298043-5, BYT-ORB1298043-50, BYT-ORB1298043-500
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
Smad, TGFbetaR1, TGFbetaRI IN 3, TGFbetaRIIN3, TGFbetaRI-IN-3, TGFb, TGF-b/Smad, TGFbRI-IN-3, TGFbetaRI-IN-3, TGF-beta/Smad, TGFbeta, TGF-beta, TGFbeta, TGFbeta/Smad
Produktbeschreibung
TGFbetaRI-IN-3 is a potent and highly selective TGFbetaR1 inhibitor (IC50 = 0.79 nM) with >2000-fold selectivity over MAP4K4. This tool compound is valuable for immuno-oncology research, enabling the study of TGF-beta signaling in both cellular assays and in vivo models of cancer and fibrosis.
Produkteigenschaften
Molekulargewicht:
465.57
Reinheit:
99.85% (May vary between batches)
CAS Nummer:
[2763602-67-9]
Formel:
C28H23N3O2S
Target-Kategorie:
TGF-beta/Smad
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: DMSO:50 mg/mL (107.4 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.3 mM)