This small molecule is a selective inhibitor of the human Bromodomain-containing protein 4 (BRD4). It is a useful chemical probe for studying BRD4 function in epigenetic regulation, cancer biology, and inflammation through in vitro biochemical and cellular assays.
Molekulargewicht:
253.34
Reinheit:
99.86% (May vary between batches)
CAS Nummer:
[218934-50-0]
Formel:
C17H19NO
Target-Kategorie:
Epigenetic Reader Domain
Anwendungsbeschreibung:
Solubility: DMSO:22.5 mg/mL (88.81 mM)
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