LML134, CAS [[1542135-76-1]]

Artikelnummer: BYT-ORB1298866
Artikelname: LML134, CAS [[1542135-76-1]]
Artikelnummer: BYT-ORB1298866
Hersteller Artikelnummer: orb1298866
Alternativnummer: BYT-ORB1298866-1, BYT-ORB1298866-1, BYT-ORB1298866-10, BYT-ORB1298866-100, BYT-ORB1298866-200, BYT-ORB1298866-25, BYT-ORB1298866-5, BYT-ORB1298866-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: H3 receptor, Histamine Receptor, HistamineReceptor, Inhibitor, LML 134, LML134, LML-134, inhibit
LML134 (LML-134) is a potent and selective inverse agonist of the human Histamine H3 Receptor (H3R), demonstrating high affinity with Kis of 0.3 nM in cAMP assays and 12 nM in binding assays. This small molecule is a valuable research tool for investigating H3R function in neurological disorders, supporting both in vitro mechanistic studies and in vivo preclinical research.
Molekulargewicht: 375.47
Reinheit: 99.86% (May vary between batches)
CAS Nummer: [1542135-76-1]
Formel: C19H29N5O3
Target-Kategorie: Histamine Receptor
Anwendungsbeschreibung: Solubility: DMSO:7.5 mg/mL (19.97 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.66 mM)