Temuterkib, CAS [[1951483-29-6]]
Artikelnummer:
BYT-ORB1303171
Produktübersicht
Artikelname:
Temuterkib, CAS [[1951483-29-6]]
Artikelnummer:
BYT-ORB1303171
Hersteller Artikelnummer:
orb1303171
Alternativnummer:
BYT-ORB1303171-1, BYT-ORB1303171-1, BYT-ORB1303171-10, BYT-ORB1303171-100, BYT-ORB1303171-2, BYT-ORB1303171-25, BYT-ORB1303171-5, BYT-ORB1303171-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
inhibit, LY3214996, LY-3214996, LY 3214996, Inhibitor, ERK1, ERK2, ERK, Extracellular signal regulated kinases, Temuterkib
Produktbeschreibung
Temuterkib (LY3214996) is an oral, potent, and selective ERK1/2 inhibitor with antineoplastic potential. It is used in cancer research, particularly for studying MAPK pathway-driven tumors, and has demonstrated activity in both in vitro cellular assays and in vivo xenograft models.
Produkteigenschaften
Molekulargewicht:
453.56
Reinheit:
>99.99% (May vary between batches)
CAS Nummer:
[1951483-29-6]
Formel:
C22H27N7O2S
Target-Kategorie:
ERK
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: DMSO:7.36 mg/mL (16.23 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.2 mM),H2O:< 1 mg/mL (insoluble or slightly soluble)