ETC-159, CAS [[1638250-96-0]]
Artikelnummer:
BYT-ORB1303253
Produktübersicht
Artikelname:
ETC-159, CAS [[1638250-96-0]]
Artikelnummer:
BYT-ORB1303253
Hersteller Artikelnummer:
orb1303253
Alternativnummer:
BYT-ORB1303253-1, BYT-ORB1303253-10, BYT-ORB1303253-100, BYT-ORB1303253-25, BYT-ORB1303253-5, BYT-ORB1303253-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
beta-catenin, betacatenin, bcatenin, Inhibitor, ETC 159, ETC 1922159, ETC159, ETC-159, ETC1922159, ETC-1922159, inhibit, Porcupine, Porcn, Wnt, Wnt/b-catenin, Wnt/betacatenin, Wnt/beta-catenin, betacatenin, beta-catenin
Produktbeschreibung
ETC-159 is a potent and orally bioavailable small molecule inhibitor of PORCN, demonstrating an IC50 of 2.9 nM in beta-catenin pathway reporter assays. It is a valuable research tool for investigating Wnt/beta-catenin signaling in various cancer models, both in vitro and in vivo.
Produkteigenschaften
Molekulargewicht:
391.38
Reinheit:
99.40% (May vary between batches)
CAS Nummer:
[1638250-96-0]
Formel:
C19H17N7O3
Target-Kategorie:
Porcupine,Wnt/beta-catenin
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.11 mM),DMSO:55 mg/mL (140.53 mM)