MRTX-1719, CAS [[2630904-45-7]]

Artikelnummer: BYT-ORB1303284
Artikelname: MRTX-1719, CAS [[2630904-45-7]]
Artikelnummer: BYT-ORB1303284
Hersteller Artikelnummer: orb1303284
Alternativnummer: BYT-ORB1303284-1, BYT-ORB1303284-1, BYT-ORB1303284-10, BYT-ORB1303284-25, BYT-ORB1303284-5, BYT-ORB1303284-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: CRC, Histone Methyltransferase, HistoneMethyltransferase, Inhibitor, inhibit, MRTX1719, MRTX-1719, MRTX 1719, MTA, NSCLC, PRMT5
MRTX-1719 is a highly potent and selective small molecule inhibitor of the PRMT5-MTA complex, demonstrating sub-10 nM IC50 activity in relevant cellular models. Its application facilitates research in oncology, particularly for investigating MTAP-deleted cancers in both in vitro and in vivo experimental settings.
Molekulargewicht: 464.88
Reinheit: 99.18% (May vary between batches)
CAS Nummer: [2630904-45-7]
Formel: C23H18ClFN6O2
Target-Kategorie: Histone Methyltransferase
Anwendungsbeschreibung: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.3 mM),DMSO:83.33 mg/mL (179.25 mM)