Pyr6, CAS [[245747-08-4]]
Artikelnummer:
BYT-ORB1307828
Produktübersicht
Artikelname:
Pyr6, CAS [[245747-08-4]]
Artikelnummer:
BYT-ORB1307828
Hersteller Artikelnummer:
orb1307828
Alternativnummer:
BYT-ORB1307828-1,BYT-ORB1307828-10,BYT-ORB1307828-25,BYT-ORB1307828-5,BYT-ORB1307828-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
Inhibitor, N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide, Pyr 6, Pyr6, Pyr-6, inhibit, Transient receptor potential channels, TRP Channel, TRPC3, TRPChannel, TRPVChannel, TRPV Channel
Produktbeschreibung
Pyr6 is a selective TRPC3 channel inhibitor with an IC50 of 0.49 µM, demonstrating higher potency against CRAC-mediated calcium entry. This compound is a valuable research tool for studying receptor-operated calcium signaling in cellular models, including mast cell and immune cell research.
Produkteigenschaften
Molekulargewicht:
418.27
Reinheit:
99.18% (May vary between batches)
CAS Nummer:
[245747-08-4]
Formel:
C17H9F7N4O
Target-Kategorie:
Calcium Channel,TRP/TRPV Channel
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:10 mg/mL (23.91 mM),DMSO:95 mg/mL (227.13 mM)