ARN14988 is a potent acid ceramidase inhibitor (human enzyme IC50 = 12.8 nM). It elevates C16 ceramide species in multiple melanoma cell lines and demonstrates anti-proliferative effects, supporting its use in cancer research, particularly for studying ceramide metabolism in vitro.
Molekulargewicht:
373.83
CAS Nummer:
[1502027-70-4]
Formel:
C16H24ClN3O5
Target-Kategorie:
Others
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