Tarafenacin is a potent and highly selective antagonist of the M3 muscarinic receptor (Ki = 0.19 nM), exhibiting approximately 200-fold selectivity versus the M2 subtype. This profile makes it a valuable research tool for investigating M3 receptor function in vitro and in vivo, particularly in studies of smooth muscle contraction and secretory processes.
Molekulargewicht:
408.39
CAS Nummer:
[385367-47-5]
Formel:
C21H20F4N2O2
Target-Kategorie:
AChR,Others
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