Radequinil is a benzodiazepine receptor partial inverse agonist with high affinity for both GABA(-) and GABA(+) ligand binding sites (Kis: 5.15 and 6.11 nM). It is a valuable research tool for investigating GABA_A receptor function in neurological studies, applicable in both in vitro binding assays and in vivo behavioral models.
Molekulargewicht:
334.33
CAS Nummer:
[219846-31-8]
Formel:
C18H14N4O3
Target-Kategorie:
GABA Receptor
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