GSK3368715 dihydrochloride, CAS [[1628925-77-8]]

Artikelnummer: BYT-ORB1709523
Artikelname: GSK3368715 dihydrochloride, CAS [[1628925-77-8]]
Artikelnummer: BYT-ORB1709523
Hersteller Artikelnummer: orb1709523
Alternativnummer: BYT-ORB1709523-1,BYT-ORB1709523-5
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: Histone Methyltransferase, HistoneMethyltransferase, GSK 3368715, GSK 3368715 Dihydrochloride, GSK3368715, GSK-3368715, GSK3368715 2HCl, GSK3368715 Dihydrochloride, GSK-3368715 Dihydrochloride, EPZ019997, EPZ-019997, EPZ019997 2HCl, EPZ019997 dihydrochloride, EPZ-019997 Dihydrochloride, EPZ 019997 Dihydrochloride, EPZ 019997, PRMT8, PRMT4, PRMT6, PRMT3, PRMT1
GSK3368715 dihydrochloride is a potent, orally bioavailable pan-inhibitor of type I PRMT enzymes (PRMT1, 3, 4, 6, 8). It exhibits anticancer activity and is a valuable chemical probe for investigating PRMT biology in both cellular assays and in vivo models of advanced solid tumors.
Molekulargewicht: 439.46
Reinheit: 99.66% (May vary between batches)
CAS Nummer: [1628925-77-8]
Formel: C20H40Cl2N4O2
Target-Kategorie: Histone Methyltransferase
Anwendungsbeschreibung: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.1 mM),H2O:100 mg/mL (227.55 mM),DMSO:100 mg/mL (227.55 mM)