GSK3368715 dihydrochloride, CAS [[1628925-77-8]]
Artikelnummer:
BYT-ORB1709523
Produktübersicht
Artikelname:
GSK3368715 dihydrochloride, CAS [[1628925-77-8]]
Artikelnummer:
BYT-ORB1709523
Hersteller Artikelnummer:
orb1709523
Alternativnummer:
BYT-ORB1709523-1,BYT-ORB1709523-5
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
Histone Methyltransferase, HistoneMethyltransferase, GSK 3368715, GSK 3368715 Dihydrochloride, GSK3368715, GSK-3368715, GSK3368715 2HCl, GSK3368715 Dihydrochloride, GSK-3368715 Dihydrochloride, EPZ019997, EPZ-019997, EPZ019997 2HCl, EPZ019997 dihydrochloride, EPZ-019997 Dihydrochloride, EPZ 019997 Dihydrochloride, EPZ 019997, PRMT8, PRMT4, PRMT6, PRMT3, PRMT1
Produktbeschreibung
GSK3368715 dihydrochloride is a potent, orally bioavailable pan-inhibitor of type I PRMT enzymes (PRMT1, 3, 4, 6, 8). It exhibits anticancer activity and is a valuable chemical probe for investigating PRMT biology in both cellular assays and in vivo models of advanced solid tumors.
Produkteigenschaften
Molekulargewicht:
439.46
Reinheit:
99.66% (May vary between batches)
CAS Nummer:
[1628925-77-8]
Formel:
C20H40Cl2N4O2
Target-Kategorie:
Histone Methyltransferase
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.1 mM),H2O:100 mg/mL (227.55 mM),DMSO:100 mg/mL (227.55 mM)