Molibresib besylate, CAS [[1895049-20-3]]

Artikelnummer: BYT-ORB1709549
Artikelname: Molibresib besylate, CAS [[1895049-20-3]]
Artikelnummer: BYT-ORB1709549
Hersteller Artikelnummer: orb1709549
Alternativnummer: BYT-ORB1709549-2
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: BET, I-BET 762 besylate, GSK 525762C, EpigeneticReaderDomain, Epigenetic Reader Domain, Molibresib besylate, ROS
Molibresib besylate (GSK525762C) is a potent and selective BET bromodomain inhibitor studied for refractory hematologic cancers. It induces reactive oxygen species (ROS) and ATM activation, demonstrating antitumor activity in both in vitro and in vivo preclinical models.
Molekulargewicht: 582.07
Reinheit: 99.64% (May vary between batches)
CAS Nummer: [1895049-20-3]
Formel: C28H28ClN5O5S
Target-Kategorie: ROS,Epigenetic Reader Domain
Anwendungsbeschreibung: Solubility: DMSO:20 mg/mL (34.36 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.44 mM)