GNA002 is a covalent and highly selective small molecule inhibitor of EZH2 with an IC50 of 1.1 µM. It is a valuable chemical probe for investigating the role of EZH2-mediated histone methylation in oncology and epigenetics research, applicable in both cellular and animal studies.
Molekulargewicht:
701.89
CAS Nummer:
[1385035-79-9]
Formel:
C42H55NO8
Target-Kategorie:
Histone Methyltransferase
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