PBRM1-BD2-IN-1 is a cell-permeable, selective inhibitor of the PBRM1 bromodomain 2 (BD2) with a Kd of 0.7 µM and an IC50 of 0.2 µM. It is a valuable chemical probe for investigating the role of PBRM1 in oncology, supporting both in vitro biochemical assays and cellular mechanism-of-action studies.
Molekulargewicht:
302.8
CAS Nummer:
[1915012-21-3]
Formel:
C17H19ClN2O
Target-Kategorie:
Others,Epigenetic Reader Domain
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