SJ995973, CAS [[2882065-25-8]]

Artikelnummer: BYT-ORB2279015
Artikelname: SJ995973, CAS [[2882065-25-8]]
Artikelnummer: BYT-ORB2279015
Hersteller Artikelnummer: orb2279015
Alternativnummer: BYT-ORB2279015-1,BYT-ORB2279015-10,BYT-ORB2279015-25,BYT-ORB2279015-5,BYT-ORB2279015-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: PROTAC, SJ 995973, SJ-995973
SJ995973 is a potent and selective BET PROTAC degrader. It induces targeted degradation of BET proteins, demonstrating robust anti-proliferative activity in cancer cell lines and promising efficacy in xenograft models, making it a valuable chemical probe for oncology and epigenetics research.
Molekulargewicht: 730.28
Reinheit: 99.36% (May vary between batches)
CAS Nummer: [2882065-25-8]
Formel: C37H40ClN7O5S
Target-Kategorie: PROTACs
Anwendungsbeschreibung: Solubility: DMSO:80 mg/mL (109.55 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (4.52 mM)