LDHA-IN-9 (Compound 1g) is a potent LDH-A inhibitor with an IC50 of 25 nM. It demonstrates anti-proliferative effects in DLD-1 cells (GI50 27 µM) via apoptosis induction and shows in vivo antitumor activity at 25 mg/kg in mouse models with minimal toxicity, supporting its use in cancer metabolism research.
Molekulargewicht:
384.27
CAS Nummer:
[862719-04-8]
Formel:
C17H22BrNO4
Target-Kategorie:
Apoptosis,Dehydrogenase
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