Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage

Produktübersicht

• Artikelname: Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage
• Artikelnummer: BYT-ORB3136482
• Hersteller Artikelnummer: orb3136482
• Alternativnummer: BYT-ORB3136482-10, BYT-ORB3136482-50
• Hersteller: Biorbyt
• Kategorie: Biochemikalien

Produktbeschreibung

Dopamine D3 receptor antagonist-3 is a selective positive allosteric modulator-antagonist (PAM-antagonist) of the D3 dopamine receptor (D3R) that can cross the blood-brain barrier. It demonstrates antagonistic activity in D3R-mediated beta-arrestin recruitment assays with an IC50 of 2.5 µM and Kb of 0.49 µM, and in D3R-mediated Go-BRET assays with an IC50 of 0.34 µM. Dopamine D3 receptor antagonist-3 is applicable for the study of neuropsychiatric disorders, including substance use disorders.

Produkteigenschaften

• Molekulargewicht: 485.86
• CAS Nummer: [2894793-37-2]
• Formel: C18H17ClF5N3O3S
• Target-Kategorie: Dopamine Receptor