WEB-2086, CAS [[105219-56-5]]

Artikelnummer: FBM-10-1389
Artikelname: WEB-2086, CAS [[105219-56-5]]
Artikelnummer: FBM-10-1389
Hersteller Artikelnummer: 10-1389
Alternativnummer: FBM-10-1389-1MG, FBM-10-1389-5MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: Chemical Name: 4-[3-[4[(2-Chlorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a]diazepin-2-yl]-1-oxopropyl]morpholine. Alternate Names: Apafant
PAF receptor antagonist
Molekulargewicht: 455.96
Reinheit: 98% by TLC, NMR (Conforms)
Formulierung: White solid
CAS Nummer: [105219-56-5]
Formel: C22H22ClN5O2S
Anwendungsbeschreibung: Potent and selective antagonist of the platelet activating factor (PAF) receptor (Ki = 16.3 nM)1. Displays an activity profile which includes antiinflamatory, antiangiogenesis and anticancer activity2. Along with leukotriene antagonists, cooperatively provides a robust anti-inflammatory effect regulating PMNL migration and edema formation3. Displays analgesic effects in animal models of neuropathic pain4. Active in vivo.