ML204, CAS [[5465-86-1]]

Artikelnummer: FBM-10-2841
Artikelname: ML204, CAS [[5465-86-1]]
Artikelnummer: FBM-10-2841
Hersteller Artikelnummer: 10-2841
Alternativnummer: FBM-10-2841-5MG, FBM-10-2841-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: Chemical Name: 4-Methyl-2-(1-piperidinyl)quinoline
TRPC4 blocker
Molekulargewicht: 226.32
Reinheit: 98% by TLC, NMR (Conforms)
Formulierung: Off-white solid
CAS Nummer: [5465-86-1]
Formel: C15H18N2
Anwendungsbeschreibung: Selective blocker of TRPC4 channels (IC50 = 0.96 - 2.6 µM, depending on assay). Displays 19-fold selectivity against TRPC6 and 9-fold selectivity against TRPC5. Has no significant activity at TRPV1, TRPV3, TRPA1 and TRPM8 channels at concentrations up to 22 µM. A useful tool for exploring the involvement of TRPC and TRPC-like channels in cellular signaling and physiology.2-4