BAY-1797, CAS [[2055602-83-8]]
Artikelnummer:
FBM-10-3980
| Artikelname: |
BAY-1797, CAS [[2055602-83-8]] |
| Artikelnummer: |
FBM-10-3980 |
| Hersteller Artikelnummer: |
10-3980 |
| Alternativnummer: |
FBM-10-3980-5MG,FBM-10-3980-25MG |
| Hersteller: |
Focus Biomolecules |
| Kategorie: |
Biochemikalien |
| Molekulargewicht: |
416.88 |
| Reinheit: |
98% by HPLC , NMR (Conforms) |
| Formulierung: |
Pale brown solid |
| CAS Nummer: |
[2055602-83-8] |
| Formel: |
C20H17ClN2O4S |
| Anwendungsbeschreibung: |
BAY-1797 (2055602-83-8) is a selective P2X4 receptor antagonist (IC50 = 211 nM HEK cellular assay, P2X4 calcium influx based assays - hIC50 = 108 nM, mIC50 = 112 nM, rIC50 = 233 nM).1 Displayed antinociceptive and anti-inflammatory effects in mouse CFA inflammatory pain models. |