Chemical Name: 4-[(2,6-Dichlorobenzoyl)amino]-N-piperidin-4-yl-1H-pyrazole-5-carboxamide hydrochloride
CDK inhibitor
Molekulargewicht:
418.70
Reinheit:
>98% by HPLC NMR (Conforms)
Formulierung:
White solid
CAS Nummer:
[902135-91-5]
Formel:
C16H17Cl2N5O2HCl
Anwendungsbeschreibung:
AT7519 is a potent CDK inhibitor. Inhibits CDKs 1,2,4,5,6, and 9 (IC50s respectively: 210 nM, 47 nM, 100 nM, 13 nM, 170 nM, and <10 nM).1,2 Active in multiple human cancer cell lines.3-7 AT7519 has also been found to be a human RORgammat agonist.8
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