PAP-1 (Standard), CAS [[870653-45-5]] Preis auf Anfrage

Artikelnummer: MCE-HY-10015R
Artikelname: PAP-1 (Standard), CAS [[870653-45-5]] Preis auf Anfrage
Artikelnummer: MCE-HY-10015R
Hersteller Artikelnummer: HY-10015R
Alternativnummer: MCE-HY-10015R-5MG, MCE-HY-10015R-1MG, MCE-HY-10015R-10MG, MCE-HY-10015R-50MG, MCE-HY-10015R-100MG, MCE-HY-10015R-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: 5-(4-Phenoxybutoxy)psoralen (Standard)
PAP-1 (Standard) is the analytical standard of PAP-1. This product is intended for research and analytical applications. PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a potent, selective, and orally active Kv1.3 blocker (EC50=2 nM). PAP-1 blocks Kv1.3 in a use-dependent manner and acts by preferentially binding to the C-type inactivated state of the channel. PAP-1 exhibits 23-fold selectivity over Kv1.5 (EC50=45 nM), and further displays 33- to 125-fold selectivity over all other Kv1-family channels. PAP-1 does not exhibit cytotoxic or phototoxic effects[1][2].
Molekulargewicht: 350.36
CAS Nummer: [870653-45-5]
Formel: C21H18O5
Target-Kategorie: Potassium Channel,Reference Standards
Anwendungsbeschreibung: Reference Standards