Varenicline-15N,13C,d2 Preis auf Anfrage

Produktübersicht

• Artikelname: Varenicline-15N,13C,d2 Preis auf Anfrage
• Artikelnummer: MCE-HY-10019S1
• Hersteller Artikelnummer: HY-10019S1
• Alternativnummer: MCE-HY-10019S1-1MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: CP 526555-15N,13C,d2

Produktbeschreibung

Varenicline-15N,13C,d2 is 15N and deuterated labeled Varenicline (HY-10019). Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50=250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agonist of alpha7beta2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].

Produkteigenschaften

• Molekulargewicht: 215.26
• Formel: C12 13CH11D2N2 15N
• Target-Kategorie: Isotope-Labeled Compounds,nAChR

Anwendungsbeschreibung

• Anwendungsbeschreibung: Isotope-Labeled Compounds