Varenicline-13C15N, CAS [[2140265-12-7]] Preis auf Anfrage

Artikelnummer: MCE-HY-10019S2
Artikelname: Varenicline-13C15N, CAS [[2140265-12-7]] Preis auf Anfrage
Artikelnummer: MCE-HY-10019S2
Hersteller Artikelnummer: HY-10019S2
Alternativnummer: MCE-HY-10019S2-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: CP 526555-13C15N
Varenicline-13C15N (CP 526555-13C15N) is 13C and 15N labeled Varenicline. Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agonist of alpha7beta2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].
Molekulargewicht: 213.22
CAS Nummer: [2140265-12-7]
Formel: C11 13C2H11N 15N2
Target-Kategorie: Isotope-Labeled Compounds,nAChR
Anwendungsbeschreibung: Isotope-Labeled Compounds