Varenicline-15N3 (hydrochloride), CAS [[1244134-80-2]] Preis auf Anfrage

Produktübersicht

• Artikelname: Varenicline-15N3 (hydrochloride), CAS [[1244134-80-2]] Preis auf Anfrage
• Artikelnummer: MCE-HY-10020S
• Hersteller Artikelnummer: HY-10020S
• Alternativnummer: MCE-HY-10020S-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: CP 526555-15N3 (Hydrochloride)

Produktbeschreibung

Varenicline-15N3 Hydrochloride (CP 526555-15N3 Hydrochloride) is the 15N labeled isotope of Varenicline hydrochloride (HY-10020). Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agonist of alpha6beta2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].

Produkteigenschaften

• Molekulargewicht: 250.70
• CAS Nummer: [1244134-80-2]
• Formel: C13H14Cl 15N3
• Target-Kategorie: Isotope-Labeled Compounds,nAChR

Anwendungsbeschreibung

• Anwendungsbeschreibung: Isotope-Labeled Compounds