MRK-016, CAS [[342652-67-9]]

Produktübersicht

• Artikelname: MRK-016, CAS [[342652-67-9]]
• Artikelnummer: MCE-HY-100370
• Hersteller Artikelnummer: HY-100370
• Alternativnummer: MCE-HY-100370-10MMX1ML,MCE-HY-100370-50MG,MCE-HY-100370-25MG,MCE-HY-100370-5MG,MCE-HY-100370-10MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

MRK-016 is a selective, orally bioavailable inverse agonist of GABAA alpha5 receptor, with an EC50 of 3 nM for GABAA alpha5, and Kis of 0.83, 0.85, 0.77 and 1.4 nM for human GABAA alpha1beta3gamma2, GABAA alpha2beta3gamma2, GABAA alpha3beta3gamma2, and GABAA alpha5beta3gamma2, respectively, MRK-016 also readily penetrates the CNS.

Produkteigenschaften

• Molekulargewicht: 368.39
• Reinheit: 99.71
• CAS Nummer: [342652-67-9]
• Formel: C17H20N8O2
• Target-Kategorie: GABA Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: Reference compound