LOC14, CAS [[877963-94-5]]

Artikelnummer: MCE-HY-100432
Artikelname: LOC14, CAS [[877963-94-5]]
Artikelnummer: MCE-HY-100432
Hersteller Artikelnummer: HY-100432
Alternativnummer: MCE-HY-100432-100MG,MCE-HY-100432-50MG,MCE-HY-100432-5MG,MCE-HY-100432-10MG,MCE-HY-100432-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
LOC14 is a potent Protein disulfide isomerase (PDI) inhibitor with EC50 and Kd values of 500 nM and 62 nM, respectively. LOC14 exhibits high stability in mouse liver microsomes and blood plasma, low intrinsic microsome clearance, and low plasma-protein binding[1]. LOC14 inhibits PDIA3 activity, decreases intramolecular disulfide bonds and subsequent oligomerization (maturation) of HA in lung epithelial cells[3].
Molekulargewicht: 317.41
Reinheit: 98
CAS Nummer: [877963-94-5]
Formel: C16H19N3O2S
Target-Kategorie: PDI
Anwendungsbeschreibung: Reference compound