EED226, CAS [[2083627-02-3]]

Produktübersicht

• Artikelname: EED226, CAS [[2083627-02-3]]
• Artikelnummer: MCE-HY-101117
• Hersteller Artikelnummer: HY-101117
• Alternativnummer: MCE-HY-101117-10MG,MCE-HY-101117-5MG,MCE-HY-101117-100MG,MCE-HY-101117-10MMX1ML,MCE-HY-101117-25MG,MCE-HY-101117-50MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

EED226 is a polycomb repressive complex 2 (PRC2) inhibitor, which binds to the K27me3-pocket on embryonic ectoderm development (EED) and shows strong antitumor activity in xenograft mice model[1]. EED226 is a potent, selective, and orally bioavailable EED inhibitor[2]. EED226 inhibits PRC2 with an IC50 of 23.4 nM when the H3K27me0 peptide is used as a substrate in the in vitro enzymatic assays[3].

Produkteigenschaften

• Molekulargewicht: 369.40
• Reinheit: 99.56
• CAS Nummer: [2083627-02-3]
• Formel: C17H15N5O3S
• Target-Kategorie: Histone Methyltransferase

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound