RSM-932A (TCD-717) is a specific ChoKalpha inhibitor with IC50s of 1 and 33 µM for human recombinant ChoKalpha and ChoKbeta enzymes, respectively. RSM-932A acts as the ''first in humans compound targeting ChoKalpha. RSM-932A is potent in vitro anti-proliferative and in vivo anti-tumoral activity against human xenografts in mice, showing high efficacy with low toxicity profiles[1][2][3].
Molekulargewicht:
877.53
Reinheit:
98.44
CAS Nummer:
[850807-63-5]
Formel:
C46H38Br2Cl2N4
Target-Kategorie:
Choline Kinase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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